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KEA1-97

Product Specifications

CAS Number

2138882-71-8

Target

Apoptosis|||Caspase

Related Pathways

Apoptosis|||Proteases/Proteasome

Purity

0.987

Bioactivity

Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 ? M) . Kea1-97 destroys the interaction between thioredoxin and caspase 3 and activates caspases without affecting the activity of thioredoxin.

Smiles

Fc1ccc(cc1)-c1ccc(Nc2nc(Cl)nc(Cl)n2)cc1

Molecular Formula

C15H9Cl2FN4

Molecular Weight

335.16

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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