What is the catalog number for BI-0115?

The catalog number for BI-0115 is T9108.

What sizes are available for BI-0115?

BI-0115 is available in the following size(s): 1 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does BI-0115 come in?

BI-0115 is available in 7 different pack sizes.

BI-0115 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures BI-0115?

BI-0115 is manufactured by Molfinity.

What is the estimated delivery time for BI-0115?

Estimated delivery time for BI-0115 is approximately 10 business day(s), depending on your location.

BI-0115

Product Specifications

CAS Number

4929-23-1

Target

Lipoxygenase

Related Pathways

Metabolism

Purity

0.9969

Bioactivity

BI-0115 is a selective small molecule inhibitor of LOX-1 that blocks cellular uptake of oxLDL. It binding triggers receptor inhibition by formation of dimers of the homodimeric ligand binding domain. The structure of LOX-1 bound to BI-0115 shows that inter-ligand interactions at the receptor interfaces are key to the formation of the receptor tetramer thereby blocking oxLDL binding.