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MGH-CP1

Product Specifications

CAS Number

896657-58-2

Target

Others|||Apoptosis

Related Pathways

Apoptosis|||Others

Purity

0.9976

Bioactivity

MGH-CP1 is a potent and selective inhibitor of TEAD palmitoylation, demonstrating dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 values of 710 nM and 672 nM, respectively.

Smiles

O=C(CSc1ncn[nH]1)Nc1ccc(cc1)C12CC3CC(CC(C3)C1)C2

Molecular Formula

C20H24N4OS

Molecular Weight

368.5

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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