GSK620
Product Specifications
CAS Number
2088410-46-0
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9988
Bioactivity
GSK620 is a pan-BD2 inhibitor, which shows an anti-inflammatory phenotype in human whole blood with excellent broad selectivity, developability, and in vivo oral pharmacokinetics.GSK620 is highly selective for the BET-BD2 family of proteins, with >200-fold selectivity over all other bromodomains. GSK620 shows an anti-inflammatory phenotype in human whole blood.
Smiles
CNC(=O)c1cc(cn(Cc2ccccc2)c1=O)C(=O)NC1CC1
Molecular Formula
C18H19N3O3
Molecular Weight
325.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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