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CD73-IN-3

Product Specifications

CAS Number

2375815-63-5

Target

CD73

Related Pathways

Immunology/Inflammation

Purity

0.9976

Bioactivity

CD73-IN-3 (LY-3475070) is a potent and selective CD73 inhibitor with an IC50 of 28 nM, and its use alone or in combination with pembrolizumab is currently being tested in patients with advanced cancer.

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[H][C@@]1(C[C@@H]1C(C)C)c1cc(nnc1C)-c1c[nH]c(=O)[nH]c1=O

Molecular Formula

C15H18N4O2

Molecular Weight

286.33

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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