GSK199
Product Specifications
CAS Number
1549811-53-1
Target
PAD
Related Pathways
Chromatin/Epigenetic
Purity
0.9944
Bioactivity
GSK199 is a selective PAD4 inhibitor (IC50 of 200 nM in the absence of calcium) .
Smiles
Cl.CCn1c(cc2cccnc12)-c1nc2cc(cc(OC)c2n1C)C(=O)N1CCC[C@@H](N)C1
Molecular Formula
C24H29ClN6O2
Molecular Weight
468.98
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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