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MS7972

Product Specifications

CAS Number

352553-42-5

Target

Epigenetic Reader Domain, MDM-2/p53

Related Pathways

Apoptosis, Chromatin/Epigenetic

Purity

0.9984

Bioactivity

MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM

Smiles

CC(=O)n1c2c(CCCC2=O)c2ccccc12

Molecular Formula

C14H13NO2

Molecular Weight

227.26

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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