BMS986260
Product Specifications
CAS Number
2001559-19-7
Target
TGF-beta/Smad
Related Pathways
Stem Cells
Purity
0.9822
Bioactivity
BMS-986260 is a selective, and orally bioavailable TGFβR1 inhibitor (IC50 = 1.6 nM) .
Smiles
C(CO)N1C(=C(N=C1)C2=CC(Cl)=C(F)C=C2)C3=NN4C(C=C3)=NC=C4C#N
Molecular Formula
C18H12ClFN6O
Molecular Weight
382.78
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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