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BMS986260

Product Specifications

CAS Number

2001559-19-7

Target

TGF-beta/Smad

Related Pathways

Stem Cells

Purity

0.9822

Bioactivity

BMS-986260 is a selective, and orally bioavailable TGF?R1 inhibitor (IC50 = 1.6 nM) .

Smiles

C(CO)N1C(=C(N=C1)C2=CC(Cl)=C(F)C=C2)C3=NN4C(C=C3)=NC=C4C#N

Molecular Formula

C18H12ClFN6O

Molecular Weight

382.78

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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