BMS-1001
Product Specifications
CAS Number
2113650-03-4
Target
PD-1/PD-L1
Related Pathways
Cell Cycle/Checkpoint, Immunology/Inflammation, Apoptosis
Purity
0.9889
Bioactivity
BMS-1001 is a potent inhibitor of PD-1/PD-L1 interaction (IC50 : 2.25 nM, in a homogenous time-resolved fluorescence binding assay) .
Smiles
CC1=CC(CN[C@H](CO)C(O)=O)=C(OCC2=CC(=CC=C2)C#N)C=C1OCC1=C(C)C(=CC=C1)C1=CC2=C(OCCO2)C=C1
Molecular Formula
C35H34N2O7
Molecular Weight
594.7
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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