JCN037
Product Specifications
CAS Number
2305154-31-6
Target
EGFR
Related Pathways
Tyrosine Kinase/Adaptors, Angiogenesis, JAK/STAT signaling
Purity
>99.99%
Bioactivity
JCN037 is potent, non-covalent and brain-penetrant inhibitor of EGFR (EGFR, p-wtEGFR and pEGFRvIII with IC50 of 2.49 nM, 3.95 nM, 4.48 nM , respectively) .
Smiles
Fc1c(Br)cccc1Nc1ncnc2cc3OCCOc3cc12
Molecular Formula
C16H11BrFN3O2
Molecular Weight
376.18
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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