Borussertib
Product Specifications
CAS Number
1800070-77-2
Target
Akt
Related Pathways
Cytoskeletal Signaling, PI3K/Akt/mTOR signaling
Purity
0.99
Bioactivity
Borussertib is a first-in-class covalent-allosteric inhibitor of protein kinase Akt, with an IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt.
Smiles
C=CC(=O)Nc1ccc2[nH]c(=O)n(C3CCN(Cc4ccc(cc4)-c4nc5cc[nH]c(=O)c5cc4-c4ccccc4)CC3)c2c1
Molecular Formula
C36H32N6O3
Molecular Weight
596.68
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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