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SR8278

Product Specifications

CAS Number

1254944-66-5

Target

REV-ERB|||Others

Related Pathways

Metabolism|||Others

Purity

0.9973

Bioactivity

SR8278 is an REV-ERB? antagonist (EC50 = 0.47 ?M), blocking activation of the receptor by the synthetic agonist GSK 4112

Smiles

CCOC(=O)C1Cc2ccccc2CN1C(=O)c1ccc(SC)s1

Molecular Formula

C18H19NO3S2

Molecular Weight

361.48

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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