USP25/28 inhibitor AZ1
Product Specifications
CAS Number
2165322-94-9
Target
DUB
Related Pathways
Ubiquitination, Cell Cycle/Checkpoint, DNA Damage/DNA Repair
Purity
0.9986
Bioactivity
USP25/28 inhibitor AZ1 is a selective, orally active and non-competitive dual ubiquitin-specific protease USP25/28 inhibitor with IC50 of 0.7 μM and 0.6 μM, respectively, and exhibits anti-inflammatory and anti-tumor effects.
Smiles
OCCNCc1cc(Br)ccc1OCc1ccc(F)c(c1)C(F)(F)F
Molecular Formula
C17H16BrF4NO2
Molecular Weight
422.21
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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