TEPP-46
Product Specifications
CAS Number
1221186-53-3
Target
PKM
Related Pathways
Metabolism
Purity
0.9965
Bioactivity
TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2) (AC50=92 nM), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity.
Smiles
Cn1c2cc(sc2c2cnn(Cc3cccc(N)c3)c(=O)c12)S(C)=O
Molecular Formula
C17H16N4O2S2
Molecular Weight
372.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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