GSK1016790A
Product Specifications
CAS Number
942206-85-1
Target
Calcium Channel, TRP/TRPV Channel
Related Pathways
Metabolism, Membrane transporter/Ion channel
Purity
0.9938
Bioactivity
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
Smiles
CC(C)C[C@H](NC(=O)c1cc2ccccc2s1)C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)c1ccc(Cl)cc1Cl
Molecular Formula
C28H32Cl2N4O6S2
Molecular Weight
655.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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