GSK-J1
Product Specifications
CAS Number
1373422-53-7
Target
Histone Demethylase
Related Pathways
Chromatin/Epigenetic
Purity
0.9967
Bioactivity
GSK-J1 is a highly potent H3K27 histone demethylase inhibitor with IC50 of 28 nM and 53 nM in cell-free assays for JMJD3 (KDM6B) and UTX (KDM6A), respectively, >10-fold selectivity over other tested demethylases.
Smiles
OC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
Molecular Formula
C22H23N5O2
Molecular Weight
389.45
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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