CPI-169 racemate
Product Specifications
CAS Number
1450655-76-1
Target
Epigenetic Reader Domain, Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9959
Bioactivity
CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
Smiles
CCS(=O)(=O)N1CCC(CC1)C(C)n1c(C)c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c2ccccc12
Molecular Formula
C27H36N4O5S
Molecular Weight
528.66
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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