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TG 100713

Product Specifications

CAS Number

925705-73-3

Target

PI3K

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.9817

Bioactivity

TG 100713 is a pan-PI3K inhibitor against PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of 50 nM, 24 nM, 165 nM and 215 nM, respectively.

Smiles

Nc1nc(N)c2nc(cnc2n1)-c1cccc(O)c1

Molecular Formula

C12H10N6O

Molecular Weight

254.25

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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