Istradefylline
Product Specifications
CAS Number
155270-99-8
Target
Adenosine Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9995
Bioactivity
Istradefylline (KW-6002) (Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials studying the treatment and basic science of Drug Abuse, Sleep Disorder, Hepatic Impairment, Parkinson's Disease, and Restless Legs Syndrome, among others.
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CN1C2=C(N(CC)C(=O)N(CC)C2=O)N=C1/C=C/C3=CC(OC)=C(OC)C=C3
Molecular Formula
C20H24N4O4
Molecular Weight
384.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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