EHT 1864 2HCl
Product Specifications
CAS Number
754240-09-0
Target
Ras, Rho
Related Pathways
Cell Cycle/Checkpoint, GPCR/G Protein, MAPK
Purity
0.9942
Bioactivity
EHT 1864 (EHT 1864 2HCl) is a Rac family GTPase inhibitor that blocks activation by direct binding to Rac1, Rac1b, Rac2, and Rac3 (Kd=40/50/60/250 nM) . EHT 1864 inhibits Rac, Ras, and Tiam-induced growth transformation of NIH-3T3 fibroblasts.
Smiles
Cl.Cl.FC(F)(F)c1ccc2c(SCCCCCOc3coc(CN4CCOCC4)cc3=O)ccnc2c1
Molecular Formula
C25H29Cl2F3N2O4S
Molecular Weight
581.47
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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