CGP 57380
Product Specifications
CAS Number
522629-08-9
Target
MNK, Apoptosis
Related Pathways
Apoptosis, MAPK
Purity
0.9989
Bioactivity
CGP 57380 (MNK1 Inhibitor) is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like kinases.
Smiles
Nc1ncnc2[nH]nc(Nc3ccc(F)cc3)c12
Molecular Formula
C11H9FN6
Molecular Weight
244.23
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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