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CGP 57380

Product Specifications

CAS Number

522629-08-9

Target

MNK, Apoptosis

Related Pathways

Apoptosis, MAPK

Purity

0.9989

Bioactivity

CGP 57380 (MNK1 Inhibitor) is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like kinases.

Smiles

Nc1ncnc2[nH]nc(Nc3ccc(F)cc3)c12

Molecular Formula

C11H9FN6

Molecular Weight

244.23

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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