EZH2-IN-9
Product Specifications
CAS Number
2700897-24-9
Target
Histone Methyltransferase, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
EZH2-IN-9 is a potent inhibitor of EZH2, which, through overexpression or mutations in the SET region (Y641F, Y641N, A687V, A677G point mutations), causes abnormal elevations in H3K27me3 and contributes to the growth and development of various tumours (e.g., breast cancer, prostate cancer, leukaemia) . EZH2-IN-9 has shown potential for cancer research.
Smiles
CC1=C2C(OC(C)(O2)[C@@H]3CC[C@@H](C(=O)N4CC(F)(F)C4)CC3)=C(Cl)C=C1C(NCC5=C(SC)C=C(C)NC5=O)=O
Molecular Formula
C28H32ClF2N3O5S
Molecular Weight
596.09
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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