BRD4 D1-IN-2
Product Specifications
Target
Epigenetic Reader Domain, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
BRD4 D1-IN-2 (compound 26) is a selective and potent inhibitor of BRD4 D1, exhibiting an IC50 value of less than 0.092 μM and a 15 nM affinity for BRD4 D1, with over 500-fold selectivity for BRD2 D1 and BRD4 D2.
Molecular Formula
C33H39F3N6O
Molecular Weight
592.7
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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