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BRD4 D1-IN-2

Product Specifications

Target

Epigenetic Reader Domain|||Others

Related Pathways

Chromatin/Epigenetic|||Others

Bioactivity

BRD4 D1-IN-2 (compound 26) is a selective and potent inhibitor of BRD4 D1, exhibiting an IC50 value of less than 0.092 ?M and a 15 nM affinity for BRD4 D1, with over 500-fold selectivity for BRD2 D1 and BRD4 D2.

Molecular Formula

C33H39F3N6O

Molecular Weight

592.7

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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