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EGFR-IN-18

Product Specifications

Target

EGFR, Others

Related Pathways

Angiogenesis, Tyrosine Kinase/Adaptors, JAK/STAT signaling, Others

Bioactivity

EGFR-IN-18 is a potent inhibitor of the enzymatic activity of the L858R/T790M/C797S mutant EGFR (4.9 nM) and is also able to reduce the enzymatic activity of wild-type EGFR (47 nM) .

Molecular Formula

C33H28N6O3S

Molecular Weight

588.68

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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