PLK1/BRD4-IN-1
Product Specifications
CAS Number
2412707-81-2
Target
Apoptosis, Androgen Receptor, c-Myc, Epigenetic Reader Domain, PLK, Others
Related Pathways
Cell Cycle/Checkpoint, Others, Endocrinology/Hormones, Apoptosis, Chromatin/Epigenetic
Bioactivity
PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM) that demonstrates significant anti-tumor efficacy in vivo.
Smiles
C(N1C=2C(N3C([C@H]1CC)=NN=C3C)=CN=C(NC4=C(OC)C=C(C(NC5CCN(C)CC5)=O)C=C4)N2)C6CCCCC6
Molecular Formula
C31H43N9O2
Molecular Weight
573.73
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
PKSH032951-01 10 µg
Recombinant Human Protachykinin-1/TAC1 Protein (His Tag)
Sign In for Pricing
View Details PKSH032951-02 50 µg
Recombinant Human Protachykinin-1/TAC1 Protein (His Tag)
Sign In for Pricing
View Details ![CD105 (ENG) Mouse Monoclonal Antibody [Clone ID: 3A9]](https://cdn.genprice.uk/products/937/68dd189a061270361e8fbe8e/imageurl/am06633su-n.webp)
AM06633SU-N 100 µL
CD105 (ENG) Mouse Monoclonal Antibody [Clone ID: 3A9]
Sign In for Pricing
View Details 