FAK-IN-2
Product Specifications
Target
FAK, Apoptosis, Others
Related Pathways
Cytoskeletal Signaling, Angiogenesis, Others, Tyrosine Kinase/Adaptors, Apoptosis
Bioactivity
FAK-IN-2 is a potent, orally active adherens spot kinase (FAK) inhibitor (IC50: 35 nM) that exhibits antitumour effects. FAK-IN-2 covalently inhibits FAK autophosphorylation in a dose-dependent manner and also inhibits tumour cell formation and migration and induces apoptosis.
Molecular Formula
C28H31ClN8O3
Molecular Weight
563.05
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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