GSK3739936
Product Specifications
CAS Number
1803444-21-4
Target
Others|||HIV Protease
Related Pathways
Proteases/Proteasome|||Microbiology/Virology|||Others
Bioactivity
GSK3739936 is a potent inhibitor of HIV-1 allosteric integrase (IC50: 11.1 nM, EC50: 1.7 nM) . GSK3739936 is also a weak inhibitor of CYP with an IC50 >24.3 ?M. It has good pharmacokinetic properties with rapid absorption, low to moderate clearance and good oral bioavailability.
Smiles
[C@@H](OC(C)(C)C)(C(O)=O)C1=C(C(=C(C)N=C1C)C2=CC=C(OCCC3=CC=C(F)C=C3)C=C2)N4CCC(C)(C)CC4
Molecular Formula
C34H43FN2O4
Molecular Weight
562.71
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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