B026
Product Specifications
CAS Number
2379416-48-3
Target
Others, Histone Acetyltransferase
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
B026 is a selective, orally active inhibitor of p300/CBP histone acetyltransferase (p300/CBP HAT) that acts on p300 (IC50: 1.8 nM) and CBP (IC50: 9.5 nM) . b026 exhibits anticancer effects on androgen receptor positive (AR+) prostate cancer cells.
Smiles
O=C1[C@]2(C=3C(CC2)=CC(=CC3)C4=CN(C)N=C4)NC(=O)N1CC(=O)N5[C@H](C(F)(F)F)COC=6C(C5)=CC(F)=CC6
Molecular Formula
C27H23F4N5O4
Molecular Weight
557.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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