DNMT3A-IN-1
Product Specifications
CAS Number
1403598-56-0
Target
Others, DNA Methyltransferase
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
DNMT3A-IN-1 is a selective and potent DNMT3A inhibitor. DNMT3A-IN-1 exhibits inhibitory activity against DNMT3A with a KI ranging from 9.16-18.85 μM (AdoMet) and 11.37-23.34 μM (poly dI-dC) .
Smiles
COc1ccc(cc1OCCCCOc1ccc(cc1)-c1nnn[nH]1)C1=NN(C2CCCCCC2)C(=O)C1(C)C
Molecular Formula
C30H38N6O4
Molecular Weight
546.66
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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