I-BET282E
Product Specifications
Target
Epigenetic Reader Domain, Others
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
I-BET282E is a pan-inhibitor of eight BET bromodomains and shows selectivity for other representative bromodomain-containing proteins. It can act on eight BRD2 (BD1/BD2), BRD2 (BD1/BD), BRD3 (BD1/BD), and BRD4 (BD1/BD), with their pIC50 values ranging from 6.4 to 7.7.
Molecular Formula
C26H34N4O7S
Molecular Weight
546.64
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog