P300 bromodomain-IN-1
Product Specifications
Target
Others, Histone Acetyltransferase, Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
P300 bromodomain-IN-1 is a potent inhibitor of p300 (EP300) bromodomain (IC50: 49 nM) . p300 bromodomain-IN-1 blocks c-Myc expression and induces cell cycle arrest at G1/G0 phase and apoptosis in OPM-2 cells. apoptosis) .
Molecular Formula
C29H31ClN4O4
Molecular Weight
535.03
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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