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A-966492

Product Specifications

CAS Number

934162-61-5

Target

PARP

Related Pathways

Chromatin/Epigenetic, DNA Damage/DNA Repair

Purity

0.9927

Bioactivity

A-96649 is a new-type and effective inhibitor. The Ki of A-966492 for PARP1 and PARP2 is 1 nM and 1.5 nM, respectively.

Smiles

NC(=O)c1cccc2[nH]c(nc12)-c1ccc(cc1F)[C@@H]1CCCN1

Molecular Formula

C18H17FN4O

Molecular Weight

324.35

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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