CCG-273463
Product Specifications
CAS Number
2750413-99-9
Target
Others, GRK
Related Pathways
GPCR/G Protein, Others
Bioactivity
CCG-273463 is a potent, covalent, selective inhibitor of GRK5 (IC50: 9 nM) . CCG-273463 can be used to study heart failure, hypertrophic cardiomyopathy and cancer.
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C(=C\1/C=2C(NC1=O)=CC=C(C(N[C@H](C)C3=CC=CC=C3)=O)C2)\C4=C(C)C(NC(CBr)=O)=C(C)N4
Molecular Formula
C26H25BrN4O3
Molecular Weight
521.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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