Glucocorticoid receptor-IN-1
Product Specifications
CAS Number
2662908-25-8
Target
Others|||Glucocorticoid Receptor|||MMP
Related Pathways
Endocrinology/Hormones|||Proteases/Proteasome|||Others
Bioactivity
Glucocorticoid receptor-IN-1 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. glucocorticoid receptor-IN-1 has good transcriptional repression, acting on hMMP1 (IC50: 2.11 nM) and also has a transcriptional activating effect on MMTV (EC50: 5.59 nM) .
Smiles
O([C@@H]([C@@H](NC(C(C)(F)F)=O)C)C1=CC(F)=CC(F)=C1)C=2C=C3C(N(N=N3)C4=CN5C(C=C4)=NN=C5)=CC2
Molecular Formula
C24H19F4N7O2
Molecular Weight
513.45
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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