GSK040
Product Specifications
CAS Number
2752331-09-0
Target
Epigenetic Reader Domain, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
GSK040, a potent and highly selective inhibitor of BET BD2, exhibits a pIC50 of 8.3, demonstrating over 5000-fold selectivity against BET BD1 (pIC50=4.6) . This compound is primarily utilized in oncology and immunology research [1].This compound is unstable in powder form and other related salt forms are recommended.
Smiles
N([C@@H](C(NC)=O)[C@@H]1CCOCC1)(C(=O)C=2C=C(C)C(=O)N(C)C2)C[C@H](C3=CC=CC=C3)C4=CC=CC=N4
Molecular Formula
C29H34N4O4
Molecular Weight
502.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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