GSK040
Product Specifications
CAS Number
2752331-09-0
Target
Epigenetic Reader Domain, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
GSK040, a potent and highly selective inhibitor of BET BD2, exhibits a pIC50 of 8.3, demonstrating over 5000-fold selectivity against BET BD1 (pIC50=4.6) . This compound is primarily utilized in oncology and immunology research [1].This compound is unstable in powder form and other related salt forms are recommended.
Smiles
N([C@@H](C(NC)=O)[C@@H]1CCOCC1)(C(=O)C=2C=C(C)C(=O)N(C)C2)C[C@H](C3=CC=CC=C3)C4=CC=CC=N4
Molecular Formula
C29H34N4O4
Molecular Weight
502.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
032531-ML750 100 µL
BLM, CT (BLM, RECQ2, RECQL3, Bloom syndrome protein, DNA helicase, RecQ-like type 2, RecQ protein-like 3) (MaxLight 750) discontinued
Sign In for Pricing
View Details 