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AHR antagonist 5 hemimaleate

Product Specifications

Target

Others|||Aryl Hydrocarbon Receptor

Related Pathways

Immunology/Inflammation|||Others

Bioactivity

AHR antagonist 5 hemimaleate is a potent antagonist (IC50 < 0.5 ?M) of the orally active aryl hydrocarbon receptor (AHR) . aHR antagonist 5 hemimaleate in combination with the detection site inhibitor anti-PD-1 exhibited inhibitory effects on tumor growth.

Molecular Formula

C29H28FN7O4

Molecular Weight

499.55

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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