CCG-273220

Product Specifications

CAS Number

2750414-35-6

Target

Others, GRK

Related Pathways

GPCR/G Protein, Others

Bioactivity

CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM) .CCG-273220 covalently binds the GRK5 subfamily-specific residue Cys474 and is more selective for GRK5 than GRK2.

Smiles

C[C@@H](NC(=O)c1ccc2NC(=O)\C(=C/c3[nH]c(C)c(NC(=O)CCl)c3C)c2c1)c1ccc(F)cc1

Molecular Formula

C26H24ClFN4O3

Molecular Weight

494.95

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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