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PDHK-IN-5

Product Specifications

Target

Others, Dehydrogenase

Related Pathways

Others, Metabolism

Bioactivity

PDHK-IN-5 is a potent inhibitor of PDHK, acting on PDHK2 (IC50: 0.006 μM) and PDHK4 (IC50: 0.0329 μM), which are drug targets for many diseases including diabetes and cancer. PDHK-IN-5 has the potential to be investigated in cancer diseases.

Molecular Formula

C30H31N5O2

Molecular Weight

493.6

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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