GRK5-IN-4

Product Specifications

CAS Number

2410794-89-5

Target

Others|||GRK

Related Pathways

GPCR/G Protein|||Others

Bioactivity

GRK5-IN-4 is a selective, potent, covalent GRK5 (G protein-coupled receptor kinase 5) inhibitor (IC50: 1.1 ?M) .GRK5-IN-4 is 90 times more selective for GRK5 than GRK2.GRK5-IN-4 can be used to study heart failure.

Smiles

N(C1=C2C(=NC(NC3=C(OC)C=C(CNC(C#CC)=O)C=C3)=N1)NC=C2)C4=C(C(NC)=O)C=CC=C4

Molecular Formula

C26H25N7O3

Molecular Weight

483.52

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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