GRK5-IN-4
Product Specifications
CAS Number
2410794-89-5
Target
Others, GRK
Related Pathways
GPCR/G Protein, Others
Bioactivity
GRK5-IN-4 is a selective, potent, covalent GRK5 (G protein-coupled receptor kinase 5) inhibitor (IC50: 1.1 μM) .GRK5-IN-4 is 90 times more selective for GRK5 than GRK2.GRK5-IN-4 can be used to study heart failure.
Smiles
N(C1=C2C(=NC(NC3=C(OC)C=C(CNC(C#CC)=O)C=C3)=N1)NC=C2)C4=C(C(NC)=O)C=CC=C4
Molecular Formula
C26H25N7O3
Molecular Weight
483.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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