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EGFR-IN-47

Product Specifications

Target

Others|||Apoptosis|||EGFR

Related Pathways

JAK/STAT signaling|||Tyrosine Kinase/Adaptors|||Angiogenesis|||Others|||Apoptosis

Bioactivity

EGFR-IN-47 is a potent, orally active inhibitor of EGFRL858R/T790M/C797S (IC50: 0.01 ?M) . EGFR-IN-47 is capable of blocking the cell cycle and inducing apoptosis. EGFR-IN-47 has potential for NSCLC studies.

Molecular Formula

C29H35N7

Molecular Weight

481.64

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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