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CARM1-IN-3 dihydrochloride

Product Specifications

Target

Others, Histone Methyltransferase

Related Pathways

Others, Chromatin/Epigenetic

Bioactivity

CARM1-IN-3 dihydrochloride (compound 17b) is a potent and selective coactivator-associated arginine methyltransferase inhibitor, targeting CARM1 with an IC50 of 0.07 μM and exhibiting minimal activity on CARM3 (IC50 > 25 μM) .

Molecular Formula

C24H34Cl2N4O2

Molecular Weight

481.46

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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