LX-039
Product Specifications
CAS Number
2135341-09-0
Target
Estrogen Receptor/ERR, Others
Related Pathways
Endocrinology/Hormones, Others
Bioactivity
LX-039 is a potent, selective, orally active estrogen receptor degrader (EC50: 2.99 nM) with antitumor effects.LX-039 has indole C-3 chloride atoms.LX-039 has good pharmacokinetic properties in mice, low clearance, high blood levels and oral exposure.
Smiles
C(=C(CC)C1=C(Cl)C=C(F)C=C1)(C2=C(Cl)C=3C(N2)=CC=CC3)C4=CC=C(C=CC(O)=O)C=C4
Molecular Formula
C27H20Cl2FNO2
Molecular Weight
480.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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