AT7867
Product Specifications
CAS Number
857531-00-1
Target
Akt, PKA, S6 Kinase
Related Pathways
Tyrosine Kinase/Adaptors, MAPK, Cytoskeletal Signaling, PI3K/Akt/mTOR signaling
Purity
0.9965
Bioactivity
AT7867 is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 values of 32 nM, 17 nM, 47 nM, 85 nM, and 20 nM, respectively, exhibiting little activity outside the AGC kinase family.
Smiles
Clc1ccc(cc1)C1(CCNCC1)c1ccc(cc1)-c1cn[nH]c1
Molecular Formula
C20H20ClN3
Molecular Weight
337.85
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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