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IDO1-IN-13

Product Specifications

Target

Others|||IDO|||Indoleamine 2,3-Dioxygenase (IDO)

Related Pathways

Others|||Metabolism

Bioactivity

IDO1-IN-13 (compound 27a) is a potent IDO1 inhibitor with an IC50 of 61.6 nM. It inhibits cell IDO1 with an EC50 of 30 nM for HeLa cells and reduces the kyn/trp ratio by 51% in SK-OV-3 xenograft tumor tissue.

Molecular Formula

C20H16BrN5O2S

Molecular Weight

470.34

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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