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PAK1-IN-1

Product Specifications

CAS Number

2485732-30-5

Target

Others, PAK

Related Pathways

Cytoskeletal Signaling, Others

Bioactivity

PAK1-IN-1 is a selective and potent inhibitor of PAK1 (IC50: 9.8 nM) . PAK1-IN-1 inhibits PAK1-associated tumour cell migration and invasion in a dose-dependent manner.

Smiles

C(NCC=1C=CN=CC1)(=O)C=2C=3C(=CC(=CC3)C4=C(Cl)C=C(C=C4)N5C(=O)C(C)=CC=C5)NN2

Molecular Formula

C26H20ClN5O2

Molecular Weight

469.92

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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